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Covalent Fragments

Covalent fragments are increasingly popular chemical probes for validation and characterization of target proteins as well as generating valuable starting points for the design of effective inhibitors and degraders. The combination of the appropriate electrophilic warhead targeting specific amino-acid residues (Cys, Lys, Thr, Tyr, Ser, His) and a relatively simple fragment-like moiety results in valuable tool compounds that can be screened in various widely adopted HTS settings. Our Covalent Fragments are “Rule of 3” (Ro3)-compliant and available for purchase either as a whole collection or by picking and choosing individual items.

Contact
Global

Ludmila Sadovenko

lsadovenko@asinex.com
North America

Mark Parisi

mparisi@asinex.com

Toll Free: +1 877 ASINEX1

Tel: +1 336 721 1617

Fax: +1 336 721 1618

N.Chestnut St., Ste.104

Winston-Salem, NC 27101

USA

Europe

Galina Afanasyeva

gafanasyeva@asinex.com

Tel: +31 (0) 203416183

Klaprozenweg 75C, 1033NN

Amsterdam, The Netherlands

Japan

Shingo Ota

sota@asinex.com

Tel: 080-3401-9097

30-2 Higashihazu, Nishio,

Aichi Japan

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